SynInnova Laboratories Inc.

SI-1905

GNE-781, 98% (HPLC)

CAS No. :

[1936422-33-1]

MDL No. :

MFCD31693834

Synonyms : 3-(7-(Difluoromethyl)-6-(1-methyl-1H-pyrazol-4-yl)-3,4-dihydroquinolin-1(2H)-yl)-N-methyl-1-(tetrahydro-2H-pyran-4-yl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridine-5(4H)-carboxamide

Price and Availability
Pack Size	Price in USD	Quantity	Availability	Shipping Status
5MG	Request Quote	- +	Back Order	Estimated to Ship on 12.28.2024
25MG	Request Quote	- +	Back Order	Estimated to Ship on 12.28.2024
100MG	Request Quote	- +	Back Order	Estimated to Ship on 12.28.2024

Note: GNE-781 is not in stock, can be available through custom synthesis. The estimated lead-time is 8-10 weeks. The product will be characterized by NMR and MS analysis. Purity (HPLC) is usually >98%. COA, QC data, SDS will be provided along with the product. For information on pricing and availability please contact us at sales@syninnova.com or submit the Bulk Quote Request. We respond promptly. Thank You!

Chemical Properties
Mol. Formula : C₂₇H₃₃F₂N₇O₂	Mol. Weight : 525.59
Appearance : Light yellow soild	Melting Point : Not available
For Laboratory research use only, not for drug, household or other uses.

Applications : GNE-781 is a highly potent and selective CBP inhibitor with an IC₅₀ of 0.94 nM in TR-FRET assay. GNE-781 also inhibits BRET and BRD4(1) with IC₅₀s of 6.2 nM and 5100 nΜ, respectively

References : Romero F. A. et al.: J. Med. Chem., 60, 9162-9183, 2017.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.

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Your request for quote will also be accepted by e-mail at sales@syninnova.com or Fax: +1 780 485 2963.

Product ID : SI-1905

Product Name : GNE-781

Note : If you do not find your required compound in our catalogue, or not commercially available, please contact us, we will assist you to get your desired molecule. We only charge if we deliver to your satisfaction.

Site is under construction and it will coming soon. Please contact us at sales@syninnova.com for COA. Thank you!

Site is under construction and it will coming soon. Please contact us at sales@syninnova.com for HNMR. Thank you!

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SI-1905

GNE-781, 98% (HPLC)

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