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SI-5103

PQR-530, >98% (HPLC)

CAS No. : 
[1927857-61-1]    
Synonyms : (S)-4-(Difluoromethyl)-5-(4-(3-methylmorpholino)-6-morpholino-1,3,5-triazin-2-yl)pyridin-2-amine

Price and Availability
Pack Size Price in USD Quantity Availability Shipping Status
5MG180.00 Back Order Estimated to Ship on 01.20.2025
10MG280.00 Back Order Estimated to Ship on 01.20.2025
25MG500.00 Back Order Estimated to Ship on 01.20.2025
50MG750.00 Back Order Estimated to Ship on 01.20.2025
100MG1150.00 Back Order Estimated to Ship on 01.20.2025
Chemical Properties
C18H23F2N7O2 407.43
Solid Not available
For Laboratory research use only, not for drug, household or other uses.
Applications : PQR-530 is a potent, ATP-competitive, orally bioavailable and brain-penetrant dual pan-PI3K/mTORC1/2 inhibitor, with a subnanomolar Kd toward PI3Kα and mTOR (0.84 and 0.33 nM, respectively). PQR-530 is a clinical candidate for the development of therapeutic agent in oncology.
References : Rageot D. et al.: Cancer Res., 77(13 Suppl), 2017; Rageot D. et al.: J. Med Chem., 62(13), 6241-6261, 2019.
Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.
Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.

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Product ID : SI-5103

Product Name : PQR-530

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