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SI-5164

Cilomilast, >98% (HPLC)

CAS No. : 
[153259-65-5]    
MDL No. : 
MFCD09033227
Synonyms : 4-Cyano-4-(3-(cyclopentyloxy)-4-methoxyphenyl)cyclohexane-1-carboxylic acid; SB-207499

Price and Availability
Pack Size Price in USD Quantity Availability Shipping Status
5MG90.00 Back Order Estimated to Ship on 01.20.2025
10MG150.00 Back Order Estimated to Ship on 01.20.2025
50MG500.00 Back Order Estimated to Ship on 01.20.2025
100MG900.00 Back Order Estimated to Ship on 01.20.2025
Chemical Properties
C20H25NO4 343.42
Solid Not available
For Laboratory research use only, not for drug, household or other uses.
Applications : Cilomilast is a potent, selective and orally active inhibitor of Phosphodiesterase 4 (PDE4), with IC50s of ~100 and 120 nM for LPDE4 and HPDE4, respectively. Cilomilast shows selectivity for PDE4 over PDE1, PDE2, PDE3 and PDE5 (IC50=74, 65, >100, and 83 µM, respectively). Cilomilast has anti-inflammatory and immunomodulatory effects and can be used for thr research of asthma and chronic obstructive pulmonary disease (COPD).
References : Griswold D. E. et al.: J. Pharmacol Exp Ther., 287(2), 705-711, 1998; Hatzelmann A. et al.: J. Pharmacol Exp Ther., 297(1), 267-279, 2001; Barnette M. S. et al.: J. Pharmacol Exp Ther., 284(1), 420-426, 1998.
Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.
Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.

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Product ID : SI-5164

Product Name : Cilomilast

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